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Biological targets
547 targets across the universe. Most are pursued by a single company — search, or start with the most-targeted below.
- CD19
- PD-1
- BCMA
- PD-L1
- CD3
- GLP-1 receptor
- HER2
- VEGF
- IL-4R
- PSMA
- CD20
- APRIL
- EGFR
- CTLA-4
- FLT3
- FXN
- BTK
- 5-HT2A
- TL1A
- BAFF
- PRAME
- WT1
- CD122
- MEK
- TSLP
- KIT
- androgen receptor
- IL-15
- KRAS
- VEGF-A
- TDP-43
- STAT6
- CD73
- dystrophin
- frataxin
- VEGF receptors
- 5-HT7
- FcRn
- menin
- Nectin-4
- KRAS G12C
- 4-1BB
- alpha-synuclein
- CLDN18.2
- FGFR3
- IKZF1
- IKZF3
- IL-17A
- IL-6
- KRAS G12D
- MRGPRX2
- TIGIT
- 5-HT1A
- amyloid beta oligomers
- DHODH
- IL-13Rα2
- ITK
- MAGE-A4
- TGF-β
- B7-H3
- GLP-1R
- mitochondrial dysfunction
- CFTR
- CSF-1R
- GBA1
- IGF-1R
- IL-2
- IL-4
- JAK1
- MAPT
- NLRP3
- tau
- 5T4
- BAG3
- CD123
- CD33
- DLL3
- DMPK
- DUX4
- FAP
- FGFR2
- GM-CSF
- HTT
- IL-33
- IL-36R
- IRAK4
- ITGB6
- MECP2
- Nrf2
- PKP2
- SERPINA1
- TNFα
- MC4R
- AXL
- MET
- 5-HT2B
- GSK-3β
- TfR1
- p53 Y220C
- telomerase
- telomere
- D2
- D3
- D4
- IL-13
- RASP
- C1q
- FASN
- GCase
- IL-15 receptor
- MER
- MT1
- MT2
- mTOR
- p38α
- RET
- TYRO3
- BAFF-R
- CD1d
- CD70
- ERK
- farnesyl transferase
- FcγRIIb
- glucan synthase
- glucocerebrosidase
- HIF prolyl hydroxylase
- HIF-PH
- IL-17F
- IL-2 receptor complex
- IL-23
- IL-2Rβ
- iNKT
- Kv7 potassium channel
- MASP-2
- nAChR α4β2
- NHE3
- NY-ESO-1
- PI3Kα RAS-binding domain
- PRLR
- PRMT5
- ribosome
- ROR1
- Survivin
- TACI
- TTR
- α4β7
- 5-HT2A receptor
- ACTH receptor
- alpha-1 adrenergic receptor
- alpha-2 adrenergic receptor
- amyloid beta
- APOE2
- APOE4
- C3d
- CCR5
- CD28
- CD40
- CD8
- CDK9
- ENPP3
- Factor H
- folate receptor alpha
- FRα
- GABA-aminotransferase
- GABA-AT
- GABAA receptor alpha-2
- GABAA receptor alpha-4
- GIP receptor
- glucagon receptor
- inflammasome pathway
- influenza
- integrin receptors
- JAK3
- KMT2A
- KRAS G12V
- KSR
- LAR family phosphatases
- MAGEA8
- mTORC1
- NAD+
- NEK7
- NMDA receptor
- Nurr1
- panKRAS
- prolactin receptor
- PTPσ
- RHEB
- SARS-CoV-2 Spike protein
- serotonin 5-HT2A receptor
- somatostatin receptor 2
- SRC
- SST2
- Tau
- YES1
- 5-HT2C
- ALK5
- amylin receptor
- angiotensin II
- angiotensin II type 1 receptor
- AV node
- AβOs
- BEST1
- beta-sarcoglycan
- BLyS
- c-KIT
- calcitonin receptor
- calcium channel
- CD276
- CD5
- CD80
- CHK1
- CHK2
- Claudin 18.2
- cMET
- CSPG
- dihydrofolate reductase
- endothelin type A receptor
- endothelin-1
- FGF23
- GIPR
- GLP-1
- glucokinase
- HBsAg
- HGF
- HPK1
- IL-18
- IL-23p19
- IL-31
- IL-4Ra
- IL-6/JAK1
- IL23p19
- kallikreins
- KCC2
- KIT D816V
- KIT exon 17
- L-type calcium channel
- labile iron
- LRRK2
- MAGEA4/8
- MAPK
- MC2R
- MEK 1
- MEK 2
- melanocortin receptor
- NaPi2b
- NLRP3 inflammasome
- NR2E3
- OX40L
- p38α MAP kinase
- p38α MAPK
- p53
- PDE5
- PDE7
- PDGF
- PDGF receptor
- PDGFR
- PKMYT1
- PlGF
- polyQ-AR
- RORA
- RXFP1
- S2R complex
- SCF
- serine protease
- SSTR2
- SSX2
- TGFβ
- thyroid hormone receptor beta
- Tissue Factor
- TNFR2
- TP53 Y220C
- TR-Beta
- transferrin receptor
- VAV1
- VEGF-B
- VEGF-C
- WEE1
- α-synuclein
- α4β7 integrin
- σ-2 receptor
- 3CL protease
- 5-HT1
- 5-HT2
- 5-HT6
- 5HT4
- A2A receptor
- ADAR
- alpha-1 antitrypsin
- alpha-7 nicotinic acetylcholine receptor
- alpha-galactosidase A
- alpha-sarcoglycan
- ANG2
- ANGPTL3
- APE1/Ref-1
- APJ
- APLNR
- AR
- ATP7B
- AβO
- B cells
- Bach1
- BCL11A
- BCL6
- BDCA2
- beta-glucuronidase
- BK virus
- BKV VP1
- Brachyury
- BRAF
- BRD4
- C1s
- C4A
- calpain-2
- cannabinoid receptors
- CAPN2
- carbonic anhydrase
- cardiac troponin T
- CASQ2
- CBD
- CBL-B
- CCR8
- CD117
- CD137
- CD18
- CD22
- CD47
- CDH3
- CDK11
- CEA
- cereblon
- CLDN6
- CNGB1
- COL4A3
- COL4A4
- COL4A5
- COL7A1
- complement factor H
- connexin 43
- CoREST
- CRF
- CRH
- CSF1
- CSPG-PTPσ
- CUG repeat expansion
- Cx43
- Cyclophilin A
- cystathionine beta-synthase
- cytomegalovirus
- delta-like ligand 3
- Delta-like ligand 3
- DMD exon 53
- DMPK mRNA
- DMPK RNA
- dopamine transporter
- DPD
- duodenal mucosa
- dysferlin
- dystrophin exon 44
- dystrophin exon 45
- dystrophin exon 51
- dystrophin exon 53
- dystrophin exon 55
- dystrophin gene exon 45
- dystrophin gene exon 51
- dystrophin gene exon 53
- E342K
- endoplasmic reticulum stress
- EpCAM
- ER
- ErbB2
- ESR1
- estrogen receptor
- exon 44
- exon 45
- exon 51
- exon 53
- exon 55
- Factor IX
- FAP-α
- fetal hemoglobin
- FGFR1
- FGFR4
- fibroblast activation protein
- FMR1
- FMRP
- G6Pase-α
- G6PC
- GAA
- GABAA α2/3
- gamma secretase
- gamma-sarcoglycan
- GAN
- GIP
- GLA
- GLUK2
- glypican 3
- GP2
- GPC3
- GRIK2
- GSPT1
- HBG1
- HBG1/2
- HBG2
- HBS1L
- HBV
- HBV core protein
- HDAC
- Hepatitis B antibodies
- hepatitis B surface antigen
- HER2/neu
- HIF-2a
- HIF-2α
- HPV
- HPV E6
- HPV E7
- huntingtin
- huntingtin gene
- hydroxychloroquine
- IFN-γ
- IFNα2b
- IGF-1
- IGHMBP2
- IKZF1/3
- IL-1
- IL-13Rα1
- IL-15R
- IL-17AA
- IL-17AF
- IL-18 binding protein
- IL-27
- IL-36
- IL-36α
- IL-36α/γ
- IL-36γ
- IL-7Rα
- INHBE
- integrin alpha v beta 6
- interferon alpha-2b
- IRF5
- ITGB2
- JAK2 V617F
- K-ATP channels
- KLK2
- KLKB1
- Kv7
- Kv7.2/3
- LAMB3
- LAMP2
- LAMP2B
- LCA5
- light chain fibrils
- LPA1R
- MASP-3
- MBNL1
- MC1R
- MERTK
- mHTT
- microdystrophin
- mineralocorticoid receptor
- mitochondrial KATP channel
- mKRAS
- MUC1
- N-protein
- NAGLU
- Nav1.2
- Nav1.6
- Nav1.7
- NKG2A
- NMDA
- NMNAT1
- NOD2
- norepinephrine transporter
- Notch pathway
- NPM1
- Nrf1
- OTC gene
- OX40
- P-Cadherin
- p38 MAP kinase alpha
- p38α kinase
- PAH
- PDE4
- phosphorylated Tau
- PI3Kα
- PKD1
- PKD2
- platelet derived growth factor
- PNPLA3
- polyclonal antibodies
- polyglutamine-expanded androgen receptor
- potassium and hyperpolarization-activated cyclic nucleotide-gated voltage gated ion channels
- PPAR-delta
- Protein Tyrosine Kinase 7
- PSA
- PTK7
- PVRIG
- R408W
- R83C
- RAGE
- RAS
- Rb-E2F pathway
- RBM20
- RDH12
- rhNAGLU
- RHO
- RSV L-protein
- RSV N-protein
- RSV neutralizing antibodies
- RYR2
- S. pneumoniae antibodies
- sclerostin
- serotonin receptor
- serotonin transporter
- sGC
- SGSH
- SIRPα
- SIRT6
- SMARCA2
- SN38
- SNP3
- SOD1
- soluble guanylate cyclase
- STEAP1
- SUR2B
- tau mRNA
- TF
- THR-β
- TIE-2
- tissue factor
- TLR2
- TLR7
- TLR8
- TNFa
- TNNI3
- TNNT2
- TP53
- troponin C
- troponin I
- TXK
- TYK2
- tyrosine kinase
- UBE3A antisense
- URAT1
- USP1
- VE-PTP
- VLA-4
- β2-adrenergic receptor
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