prexasertib
ACR-368 Small Molecule Target: CHK1, CHK2
Most recent annual filing: 2026-03-15
Generative Phosphoproteomics Acrivon Predictive Precision Proteomics platform — quantifies compound-specific, drug-regulated pathway activity levels inside the intact cell via MS-based proteomic profiling and automated tumor imaging biomarker platform; applied to oncology drug discovery, patient selection (OncoSignature tests), indication finding, and resistance mechanism identification
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